Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with Target = 'Sodium- and chloride-dependent GABA transporter 2' and Ligand = 'BDBM90787'
TargetSodium- and chloride-dependent GABA transporter 2(Rat)
Synaptic Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 90787BDBM90787(SMR000326834 | cid_11957555 | GUVACINE | MLS000859...)
Affinity DataIC50: 5.80E+4nMAssay Description:Inhibitory activity against rat GABA transporter-2 (rGAT2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 2(Human)
Zentrum F£R Pharmaforschung

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 90787BDBM90787(SMR000326834 | cid_11957555 | GUVACINE | MLS000859...)
Affinity DataIC50: 6.60E+4nMAssay Description:Binding affinity to GAT2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 2(Mouse)
University of Louvain

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 90787BDBM90787(SMR000326834 | cid_11957555 | GUVACINE | MLS000859...)
Affinity DataIC50: 7.24E+4nMAssay Description:Inhibition of mouse GAT2 mediated [3]GABA uptake expressed in HEK293 cells after 3 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed