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Found 2 Enz. Inhib. hit(s) with Target = 'Sodium-dependent dopamine transporter' and Ligand = 'BDBM50107089'
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Nida-Irp

Curated by ChEMBL
LigandPNGBDBM50107089(CHEMBL433340 | [3-((3R,5R)-3,5-Dimethyl-piperazin-...)
Affinity DataKi:  77.1nMAssay Description:Binding affinity against dopamine transporter was determined by the displacement of [3H]WIN-35428 radioligand in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Nida-Irp

Curated by ChEMBL
LigandPNGBDBM50107089(CHEMBL433340 | [3-((3R,5R)-3,5-Dimethyl-piperazin-...)
Affinity DataKi:  83nMAssay Description:Binding affinity at Dopamine transporter by displacing [3H]WIN-35428 from rat caudate putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed