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Found 2 Enz. Inhib. hit(s) with Target = 'Sodium-dependent dopamine transporter' and Ligand = 'BDBM50129592'
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Nida-Irp

Curated by ChEMBL
LigandPNGBDBM50129592(CHEMBL87841 | N-(3-(4-benzylpiperazin-1-yl)propyl)...)
Affinity DataKi:  27.6nMAssay Description:Binding affinity against dopamine transporter was determined by the displacement of [3H]WIN-35428 radioligand in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Nida-Irp

Curated by ChEMBL
LigandPNGBDBM50129592(CHEMBL87841 | N-(3-(4-benzylpiperazin-1-yl)propyl)...)
Affinity DataIC50:  29.7nMAssay Description:Displacement of [3H]WIN 35428 from DAT in Sprague-Dawley rat striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed