Found 1 Enz. Inhib. hit(s) with Target = 'Sodium-dependent dopamine transporter' and Ligand = 'BDBM50236727'
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Virginia Commonwealth University
Curated by ChEMBL
Virginia Commonwealth University
Curated by ChEMBL
Affinity DataIC50: 2.10nMAssay Description:Inhibition of DAT in Sprague-Dawley rat synaptosomes assessed as reduction in [3H]dopamine uptake by liquid scintillation counting methodMore data for this Ligand-Target Pair