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Found 3 Enz. Inhib. hit(s) with Target = 'Sodium-dependent dopamine transporter' and Ligand = 'BDBM50302907'
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50302907(2-(N-Cyclopropylamino)-3-chloropropiophenone | CHE...)
Affinity DataKi:  1.15E+3nMAssay Description:Displacement of [125I]RTI55 from cloned human DAT expressed in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50302907(2-(N-Cyclopropylamino)-3-chloropropiophenone | CHE...)
Affinity DataIC50:  265nMAssay Description:Inhibition of [3H]dopamine reuptake at human DAT expressed in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Rti International

Curated by ChEMBL
LigandPNGBDBM50302907(2-(N-Cyclopropylamino)-3-chloropropiophenone | CHE...)
Affinity DataIC50:  533nMAssay Description:Inhibition of DAT-mediated dopamine uptake in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed