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Found 4 Enz. Inhib. hit(s) with Target = 'Sodium-dependent dopamine transporter' and Ligand = 'BDBM86699'
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Duquesne University

Curated by PDSP Ki Database
LigandPNGBDBM86699(4-ARA-127)
Affinity DataKi:  1.63E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Duquesne University

Curated by PDSP Ki Database
LigandPNGBDBM86699(4-ARA-127)
Affinity DataKi:  3.30E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Duquesne University

Curated by PDSP Ki Database
LigandPNGBDBM86699(4-ARA-127)
Affinity DataIC50:  24.8nMAssay Description:Ability to displace [3H]WIN-35428 binding to dopamine transporter from rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Duquesne University

Curated by PDSP Ki Database
LigandPNGBDBM86699(4-ARA-127)
Affinity DataIC50:  85.2nMAssay Description:Inhibition of high-affinity uptake of [3H]dopamine at dopamine transporter into rat striatal nerve endings (synaptosomes)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed