Found 10 Enz. Inhib. hit(s) with Target = 'Sodium-dependent serotonin transporter' and Ligand = 'BDBM22199'
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Lundbeck Ais
Curated by PDSP Ki Database
Lundbeck Ais
Curated by PDSP Ki Database
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Lundbeck Ais
Curated by PDSP Ki Database
Lundbeck Ais
Curated by PDSP Ki Database
Affinity DataKi: 135nMAssay Description:Binding affinity against Serotonin transporter (SERT) labelled with [125I]-RTI-55 in rat.More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Lundbeck Ais
Curated by PDSP Ki Database
Lundbeck Ais
Curated by PDSP Ki Database
Affinity DataKi: 135nMAssay Description:Displacement of [125I]RTI55 from SERT in rat brain synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Lundbeck Ais
Curated by PDSP Ki Database
Lundbeck Ais
Curated by PDSP Ki Database
Affinity DataKi: 135nMAssay Description:Binding affinity towards rat serotonin transporter (SERT)More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Lundbeck Ais
Curated by PDSP Ki Database
Lundbeck Ais
Curated by PDSP Ki Database
Affinity DataKi: 140nMAssay Description:The assay was initiated by the addition of membranes to binding buffer containing test compound, blocker, and radioligand. The samples were incubated...More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Lundbeck Ais
Curated by PDSP Ki Database
Lundbeck Ais
Curated by PDSP Ki Database
Affinity DataIC50: 135nMAssay Description:Binding affinity was determined at the Serotonin transporter labeled with radioligand [125 I] RTI-55More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Lundbeck Ais
Curated by PDSP Ki Database
Lundbeck Ais
Curated by PDSP Ki Database
Affinity DataIC50: 576nMAssay Description:Reuptake inhibition of [3H]-5-HT (5-HT) in rat.More data for this Ligand-Target Pair
Affinity DataKd: 363nMAssay Description:Inhibition of [125I]RTI-55 binding to human SERT in clonal cellsMore data for this Ligand-Target Pair
Affinity DataKd: 954nMAssay Description:Inhibition of [125I]RTI-55 binding to human SERT in clonal cellsMore data for this Ligand-Target Pair
Affinity DataKd: 363nMAssay Description:Inhibition of [125I]RTI-55 binding to human SERT in clonal cellsMore data for this Ligand-Target Pair