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Found 4 Enz. Inhib. hit(s) with Target = 'Sodium-dependent serotonin transporter' and Ligand = 'BDBM50020707'
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Veterans Administration Medical Center

Curated by PDSP Ki Database
LigandPNGBDBM50020707(CHEMBL287064 | Nomelidine | Norzimelidine | [3-(4-...)
Affinity DataKi:  3.30nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Veterans Administration Medical Center

Curated by PDSP Ki Database
LigandPNGBDBM50020707(CHEMBL287064 | Nomelidine | Norzimelidine | [3-(4-...)
Affinity DataKi:  450nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Veterans Administration Medical Center

Curated by PDSP Ki Database
LigandPNGBDBM50020707(CHEMBL287064 | Nomelidine | Norzimelidine | [3-(4-...)
Affinity DataIC50:  100nMAssay Description:In vitro inhibition of accumulation of [14C]-5-HT (5-HT) in mouse brain slicesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Veterans Administration Medical Center

Curated by PDSP Ki Database
LigandPNGBDBM50020707(CHEMBL287064 | Nomelidine | Norzimelidine | [3-(4-...)
Affinity DataIC50:  100nMAssay Description:In vitro inhibition of accumulation of (-)-[3H]-Norepinephrine (NA) in mouse brain slicesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed