Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = 'Sodium-dependent serotonin transporter' and Ligand = 'BDBM50218672'
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50218672(2-(2-((dimethylamino)methyl)-4-fluorophenoxy)-5-me...)
Affinity DataKi:  7.01nMAssay Description:Displacement of [3H]paroxetine from SERT in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50218672(2-(2-((dimethylamino)methyl)-4-fluorophenoxy)-5-me...)
Affinity DataKi:  8nMAssay Description:Displacement of [3H]citalopram from human cloned SERT expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed