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Found 9 Enz. Inhib. hit(s) with Target = 'Sodium-dependent serotonin transporter' and Ligand = 'BDBM50254790'
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Mayo Clinic

Curated by PDSP Ki Database
LigandPNGBDBM50254790((S)-Norfluoxetine | CHEMBL465123 | NORFLUOXETINE)
Affinity DataKi:  1.47nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Emory University

Curated by PDSP Ki Database
LigandPNGBDBM50254790((S)-Norfluoxetine | CHEMBL465123 | NORFLUOXETINE)
Affinity DataKi:  1.90nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Mayo Clinic

Curated by PDSP Ki Database
LigandPNGBDBM50254790((S)-Norfluoxetine | CHEMBL465123 | NORFLUOXETINE)
Affinity DataKi:  2.30nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Emory University

Curated by PDSP Ki Database
LigandPNGBDBM50254790((S)-Norfluoxetine | CHEMBL465123 | NORFLUOXETINE)
Affinity DataKi:  3.15nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Emory University

Curated by PDSP Ki Database
LigandPNGBDBM50254790((S)-Norfluoxetine | CHEMBL465123 | NORFLUOXETINE)
Affinity DataKi:  3.15nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Emory University

Curated by PDSP Ki Database
LigandPNGBDBM50254790((S)-Norfluoxetine | CHEMBL465123 | NORFLUOXETINE)
Affinity DataKi:  13.9nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Mayo Clinic

Curated by PDSP Ki Database
LigandPNGBDBM50254790((S)-Norfluoxetine | CHEMBL465123 | NORFLUOXETINE)
Affinity DataKi:  50nMAssay Description:Displacement of [125I]RTI55 from human recombinant SERT expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Mayo Clinic

Curated by PDSP Ki Database
LigandPNGBDBM50254790((S)-Norfluoxetine | CHEMBL465123 | NORFLUOXETINE)
Affinity DataKi:  54nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Mayo Clinic

Curated by PDSP Ki Database
LigandPNGBDBM50254790((S)-Norfluoxetine | CHEMBL465123 | NORFLUOXETINE)
Affinity DataIC50:  46nMAssay Description:Inhibition of [3H]5HT from human recombinant SERT expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed