Found 2 Enz. Inhib. hit(s) with Target = 'Sodium-dependent serotonin transporter' and Ligand = 'BDBM50476262'
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataEC50: 2.00E+12nMAssay Description:Decrease in [3H]5-HT uptake at human SERT W103C mutant transfected in HEK293 cellsMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataEC50: 3.16E+3nMAssay Description:Decrease in [3H]5-HT uptake at human SERT G498C mutant transfected in HEK293 cellsMore data for this Ligand-Target Pair