Found 4 Enz. Inhib. hit(s) with Target = 'Sodium-dependent serotonin transporter' and Ligand = 'BDBM82219'
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Pfizer
Curated by PDSP Ki Database
Pfizer
Curated by PDSP Ki Database
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Pfizer
Curated by PDSP Ki Database
Pfizer
Curated by PDSP Ki Database
Affinity DataIC50: 840nMAssay Description:Inhibition of dopamine uptake in synaptosomal preparation in rat corpus striatum, using [3H]dopamineMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Pfizer
Curated by PDSP Ki Database
Pfizer
Curated by PDSP Ki Database
Affinity DataIC50: 1.48E+3nMAssay Description:Inhibition of 5-HT uptake in synaptosomal preparation from rat corpus striatum, using [3H]5-HTMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Pfizer
Curated by PDSP Ki Database
Pfizer
Curated by PDSP Ki Database
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of 5-HT uptake in synaptosomal preparation from rat corpus striatum, using [3H]5-HTMore data for this Ligand-Target Pair