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Found 4 Enz. Inhib. hit(s) with Target = 'Solute carrier family 15 member 1' and Ligand = 'BDBM50188516'
TargetSolute carrier family 15 member 1(Homo sapiens (Human))
Martin-Luther-University Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50188516(2-(2-amino-N-methylacetamido)acetic acid | CHEMBL1...)
Affinity DataKi:  8.30E+5nMAssay Description:Inhibition constant (Ki) for human intestinal peptide carrierMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 15 member 1(Homo sapiens (Human))
Martin-Luther-University Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50188516(2-(2-amino-N-methylacetamido)acetic acid | CHEMBL1...)
Affinity DataKi:  1.28E+7nMAssay Description:TP_TRANSPORTER: inhibition of VACV uptake in PEPT1-expressing CHO cellsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSolute carrier family 15 member 1(Homo sapiens (Human))
Martin-Luther-University Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50188516(2-(2-amino-N-methylacetamido)acetic acid | CHEMBL1...)
Affinity DataIC50:  1.16E+6nMAssay Description:Binding affinity to human PEPT1 assessed as inhibition of [14C]Gly-Sar uptake in MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 15 member 1(Homo sapiens (Human))
Martin-Luther-University Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50188516(2-(2-amino-N-methylacetamido)acetic acid | CHEMBL1...)
Affinity DataEC50:  5.40E+5nMAssay Description:Activation of human PEPT1 expressed in MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed