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Found 4 Enz. Inhib. hit(s) with Target = 'Solute carrier family 22 member 1' and Ligand = 'BDBM50420217'
TargetSolute carrier family 22 member 1(RAT)
University Of Heidelberg

Curated by ChEMBL
LigandPNGBDBM50420217(METIPRENALINE)
Affinity DataKi:  2.50E+4nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in OCT1-expressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 1(RAT)
University Of Heidelberg

Curated by ChEMBL
LigandPNGBDBM50420217(METIPRENALINE)
Affinity DataKi:  4.30E+4nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 1(RAT)
University Of Heidelberg

Curated by ChEMBL
LigandPNGBDBM50420217(METIPRENALINE)
Affinity DataIC50:  3.70E+4nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake (TEA: 10 uM) in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 1(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50420217(METIPRENALINE)
Affinity DataIC50: >1.00E+5nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake (MPP+: 0.25 uM) in OCT1-expressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed