Found 3 Enz. Inhib. hit(s) with Target = 'Solute carrier family 22 member 6' and Ligand = 'BDBM50420185'
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Nagoya University School Of Medicine
Curated by ChEMBL
Nagoya University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 2.27E+4nMAssay Description:TP_TRANSPORTER: inhibition of PAH uptake (PAH: 5 uM, indoxyl sulfate:500 uM) in S2 human-OAT1 expressing cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Nagoya University School Of Medicine
Curated by ChEMBL
Nagoya University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 2.30E+4nMAssay Description:TP_TRANSPORTER: uptake&inhibition of PAH in OAT1-S2 cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Nagoya University School Of Medicine
Curated by ChEMBL
Nagoya University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 8.30E+4nMAssay Description:TP_TRANSPORTER: inhibition of PAH uptake in OAT-expressing OK cellsMore data for this Ligand-Target Pair