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Found 3 Enz. Inhib. hit(s) with Target = 'Solute carrier family 22 member 6' and Ligand = 'BDBM50420185'
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Nagoya University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50420185(CHEMBL1233636)
Affinity DataKi:  2.27E+4nMAssay Description:TP_TRANSPORTER: inhibition of PAH uptake (PAH: 5 uM, indoxyl sulfate:500 uM) in S2 human-OAT1 expressing cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Nagoya University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50420185(CHEMBL1233636)
Affinity DataKi:  2.30E+4nMAssay Description:TP_TRANSPORTER: uptake&inhibition of PAH in OAT1-S2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Nagoya University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50420185(CHEMBL1233636)
Affinity DataIC50:  8.30E+4nMAssay Description:TP_TRANSPORTER: inhibition of PAH uptake in OAT-expressing OK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed