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Found 8 Enz. Inhib. hit(s) with Target = 'Somatostatin receptor type 2' and Ligand = 'BDBM50159392'
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50159392((4R,7R,10S,13S,16S,19S,22S,25S,28S,31S,34S,37R)-37...)
Affinity DataIC50:  2nMAssay Description:Displacement of [125I]-[Leu8, DTrp22, Tyr25]-somatostatin-28 from human recombinant sst2 receptor expressed in chinese hamster CCL39 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50159392((4R,7R,10S,13S,16S,19S,22S,25S,28S,31S,34S,37R)-37...)
Affinity DataIC50:  2.30nMAssay Description:Inhibition of [Leu8,D-Trp22,125I-Tyr25]SRIF-28 binding to human somatostatin receptor type 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50159392((4R,7R,10S,13S,16S,19S,22S,25S,28S,31S,34S,37R)-37...)
Affinity DataIC50:  2.40nMAssay Description:Displacement of [125I]-[Leu8, DTrp22, Tyr25]SRIF28 from human sst2 receptor expressed in chinese hamster CCL39 cells by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50159392((4R,7R,10S,13S,16S,19S,22S,25S,28S,31S,34S,37R)-37...)
Affinity DataIC50:  2.60nMAssay Description:Displacement of [125I]-[Leu8, DTrp22, Tyr25]SRIF-28 from human cloned sst2 receptor expressed in CCL39 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50159392((4R,7R,10S,13S,16S,19S,22S,25S,28S,31S,34S,37R)-37...)
Affinity DataIC50:  2.60nMAssay Description:Displacement of [125I]LTT-SRIF-28 from human sst2 receptor by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50159392((4R,7R,10S,13S,16S,19S,22S,25S,28S,31S,34S,37R)-37...)
Affinity DataIC50:  2.70nMAssay Description:Displacement of [125I][LTT]SRIF28 from human cloned sst2 receptor by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50159392((4R,7R,10S,13S,16S,19S,22S,25S,28S,31S,34S,37R)-37...)
Affinity DataIC50:  3nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST2 receptor expressed in human CCL39 cells by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50159392((4R,7R,10S,13S,16S,19S,22S,25S,28S,31S,34S,37R)-37...)
Affinity DataIC50:  3nMAssay Description:Displacement of [125I](Leu8,D-Trp22,Tyr25)-SRIF28 from human sst2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed