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Found 4 Enz. Inhib. hit(s) with Target = 'Somatostatin receptor type 3' and Ligand = 'BDBM50054461'
TargetSomatostatin receptor type 3(MOUSE)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50054461(CHEMBL3323073)
Affinity DataIC50:  0.700nMAssay Description:Displacement of [125I]SS-14 from mouse SSTR3 expressed in CHO cells by TopCount analyzerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50054461(CHEMBL3323073)
Affinity DataIC50:  1.5nMAssay Description:Displacement of [125I]SS-14 from human SSTR3 expressed in CHO cells by TopCount analyzerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(MOUSE)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50054461(CHEMBL3323073)
Affinity DataIC50:  3.5nMAssay Description:Antagonist activity at mouse SSTR3 expressed in CHO cells assessed as cAMP level by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50054461(CHEMBL3323073)
Affinity DataIC50:  5.40nMAssay Description:Antagonist activity at human SSTR3 expressed in CHO cells assessed as cAMP level by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed