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Found 8 Enz. Inhib. hit(s) with Target = 'Somatostatin receptor type 3' and Ligand = 'BDBM50159392'
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50159392((4R,7R,10S,13S,16S,19S,22S,25S,28S,31S,34S,37R)-37...)
Affinity DataIC50:  1.70nMAssay Description:Displacement of [125I]-[Leu8, DTrp22, Tyr25]-somatostatin-28 from human recombinant sst3 receptor expressed in chinese hamster CCL39 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50159392((4R,7R,10S,13S,16S,19S,22S,25S,28S,31S,34S,37R)-37...)
Affinity DataIC50:  2.70nMAssay Description:Displacement of [125I]-[Leu8, DTrp22, Tyr25]SRIF28 from human sst3 receptor expressed in chinese hamster CCL39 cells by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50159392((4R,7R,10S,13S,16S,19S,22S,25S,28S,31S,34S,37R)-37...)
Affinity DataIC50:  3.30nMAssay Description:Displacement of [125I][LTT]SRIF28 from human cloned sst3 receptor by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50159392((4R,7R,10S,13S,16S,19S,22S,25S,28S,31S,34S,37R)-37...)
Affinity DataIC50:  3.60nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST3 receptor expressed in human CCL39 cells by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50159392((4R,7R,10S,13S,16S,19S,22S,25S,28S,31S,34S,37R)-37...)
Affinity DataIC50:  3.60nMAssay Description:Displacement of [125I](Leu8,D-Trp22,Tyr25)-SRIF28 from human sst3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50159392((4R,7R,10S,13S,16S,19S,22S,25S,28S,31S,34S,37R)-37...)
Affinity DataIC50:  3.70nMAssay Description:Inhibition of [Leu8,D-Trp22,125I-Tyr25]SRIF-28 binding to human somatostatin receptor type 3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50159392((4R,7R,10S,13S,16S,19S,22S,25S,28S,31S,34S,37R)-37...)
Affinity DataIC50:  3.80nMAssay Description:Displacement of [125I]-[Leu8, DTrp22, Tyr25]SRIF-28 from human cloned sst3 receptor expressed in CCL39 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50159392((4R,7R,10S,13S,16S,19S,22S,25S,28S,31S,34S,37R)-37...)
Affinity DataIC50:  4.30nMAssay Description:Displacement of [125I]LTT-SRIF-28 from human sst3 receptor by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed