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Found 2 Enz. Inhib. hit(s) with Target = 'Sphingolipid delta(4)-desaturase DES1' and Ligand = 'BDBM50382314'
TargetSphingolipid delta(4)-desaturase DES1(Homo sapiens (Human))
Institute For Advanced Chemistry Of Catalonia

Curated by ChEMBL
LigandPNGBDBM50382314(CHEMBL2024680)
Affinity DataIC50:  1.81E+4nMAssay Description:Inhibition of Des1 in human A549 cells assessed as formation of CerC6NBD from dhCerC6NBD after 4 hrs by HPLC-FD analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingolipid delta(4)-desaturase DES1(Homo sapiens (Human))
Institute For Advanced Chemistry Of Catalonia

Curated by ChEMBL
LigandPNGBDBM50382314(CHEMBL2024680)
Affinity DataIC50:  1.88E+4nMAssay Description:Inhibition of Des1 in human HCT116 cells assessed as formation of CerC6NBD from dhCerC6NBD after 4 hrs by HPLC-FD analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed