TargetSphingosine kinase 1(Homo sapiens (Human))
Pennsylvania State University College Of Medicine
Curated by ChEMBL
Pennsylvania State University College Of Medicine
Curated by ChEMBL
Affinity DataKi: 1.06E+3nMAssay Description:Competitive inhibition of recombinant sphingosine kinase 1 using D-erythro-sphingosine as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
TargetSphingosine kinase 1(Homo sapiens (Human))
Pennsylvania State University College Of Medicine
Curated by ChEMBL
Pennsylvania State University College Of Medicine
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant full length GST-tagged human SPHK1 expressed in baculovirus expression system incubated for 1 hr in presence of ATP by Alex...More data for this Ligand-Target Pair