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Found 1 Enz. Inhib. hit(s) with Target = 'Steroid hormone receptor ERR1' and Ligand = 'BDBM50276833'
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL
LigandPNGBDBM50276833(CHEMBL4175927)
Affinity DataIC50:  23nMAssay Description:Antagonist activity at His6-tagged ERRalpha LBD (unknown origin) assessed as inhibition of GST-tagged SRC-2 co-activator peptide recruitment after 18...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed