Found 3 Enz. Inhib. hit(s) with Target = 'Stimulator of interferon genes protein' and Ligand = 'BDBM50587699'
TargetStimulator of interferon genes protein(Mus musculus)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 3.42E+3nMAssay Description:Antagonist activity at STING in MEF cells by Flowcytometry assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.08E+4nMAssay Description:Antagonist activity at STING in human IMR-90 cells by Flowcytometry assayMore data for this Ligand-Target Pair
Affinity DataKd: 5.30E+4nMAssay Description:Binding affinity to human NT-647-labeled C-terminal domain STING R232 mutant (149 to 379residues) expressed in Escherichia coli BL21 (DE3) assessed a...More data for this Ligand-Target Pair