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Found 3 Enz. Inhib. hit(s) with Target = 'Stromelysin-1' and Ligand = 'BDBM50082545'
TargetStromelysin-1(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50082545((S)-4-(4-Methoxy-benzenesulfonyl)-2,2-dimethyl-[1,...)
Affinity DataIC50:  0.700nMAssay Description:In vitro inhibitory activity against matrix metalloprotease-3.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50082545((S)-4-(4-Methoxy-benzenesulfonyl)-2,2-dimethyl-[1,...)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of truncated human recombinant MMP3 catalytic domain expressed in Escherichia coli BL21(DE3) after 3 hrs in presence of [H]-transferrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50082545((S)-4-(4-Methoxy-benzenesulfonyl)-2,2-dimethyl-[1,...)
Affinity DataIC50:  0.708nMAssay Description:Inhibition of MMP3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed