TargetSubstance-K receptor(Homo sapiens (Human))
Creighton University School Of Medicine
Curated by ChEMBL
Creighton University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 102nMAssay Description:The compound was tested for competition binding with [3H]NKA against the CHO cells from cloned human Tachykinin receptor 2More data for this Ligand-Target Pair
TargetSubstance-K receptor(Homo sapiens (Human))
Creighton University School Of Medicine
Curated by ChEMBL
Creighton University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 148nMAssay Description:Competitive inhibition of [125I]NKA binding to hamster urinary bladder Tachykinin receptor 2More data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Concentration required to inhibit the specific binding of [125I]NKA to Neurokinin-2 (NK-2) receptor in rat duodenum membranesMore data for this Ligand-Target Pair
TargetSubstance-K receptor(Homo sapiens (Human))
Creighton University School Of Medicine
Curated by ChEMBL
Creighton University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 245nMAssay Description:Inhibitory activity against human Tachykinin receptor 2More data for this Ligand-Target Pair
Affinity DataEC50: 167nMAssay Description:In vitro agonistic activity against tachykinin receptor 2 of rat colon muscularis mucosae.More data for this Ligand-Target Pair
Affinity DataEC50: 1nMAssay Description:Agonist activity at tachykinin receptor 2 in the rat colon muscularis mucosaeMore data for this Ligand-Target Pair
Affinity DataEC50: 167nMAssay Description:Agonist activity at tachykinin receptor 2 in the rat colon muscularis mucosaeMore data for this Ligand-Target Pair