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Found 3 Enz. Inhib. hit(s) with Target = 'Substance-P receptor' and Ligand = 'BDBM50030429'
TargetSubstance-P receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50030429(CHEMBL173396 | N-[(S)-4-(3,5-Bis-trifluoromethyl-p...)
Affinity DataIC50:  0.400nMAssay Description:Binding affinity against wild type human Tachykinin receptor 1 expressed in CHO cells was measured by its ability to displace [125I]- Tyr-8 substance...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50030429(CHEMBL173396 | N-[(S)-4-(3,5-Bis-trifluoromethyl-p...)
Affinity DataIC50:  0.5nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in CHO cells was measured by its ability to displace [125I]- Tyr-8 substance P.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50030429(CHEMBL173396 | N-[(S)-4-(3,5-Bis-trifluoromethyl-p...)
Affinity DataIC50:  10nMAssay Description:Binding affinity against Gln165Ala mutant type human Tachykinin receptor 1 expressed in CHO cells was measured by its ability to displace [125I]- Tyr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed