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Found 4 Enz. Inhib. hit(s) with Target = 'Substance-P receptor' and Ligand = 'BDBM50033817'
TargetSubstance-P receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50033817(3-(3,5-Bis-trifluoromethyl-benzyl)-5-(1H-indol-3-y...)
Affinity DataIC50:  22nMAssay Description:Binding affinity at human Tachykinin receptor 1 expressed in CHO cells by [125 I]Trp8-substance P displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50033817(3-(3,5-Bis-trifluoromethyl-benzyl)-5-(1H-indol-3-y...)
Affinity DataIC50:  22nMAssay Description:Binding affinity at human Tachykinin receptor 1 expressed in CHO cells by [125 I]Trp8-substance P displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50033817(3-(3,5-Bis-trifluoromethyl-benzyl)-5-(1H-indol-3-y...)
Affinity DataIC50:  25nMAssay Description:Antagonist activity at NK1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50033817(3-(3,5-Bis-trifluoromethyl-benzyl)-5-(1H-indol-3-y...)
Affinity DataIC50:  25.7nMAssay Description:Binding affinity was measured against the Tachykinin receptor 1 in CHO-expressed hNK1 using [125I]SP.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed