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Found 2 Enz. Inhib. hit(s) with Target = 'Substance-P receptor' and Ligand = 'BDBM50045037'
TargetSubstance-P receptor(Homo sapiens (Human))
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50045037(CHEMBL3144352 | N-Benzyl-2-[2-[2-(3,6-dioxo-2,5-di...)
Affinity DataIC50:  165nMAssay Description:Tested for antagonist activityt against NK-2 receptor in rabbit pulmonary artery by using Neurokinin A as agonistMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50045037(CHEMBL3144352 | N-Benzyl-2-[2-[2-(3,6-dioxo-2,5-di...)
Affinity DataIC50:  6.40E+3nMAssay Description:Tested for binding affinity against rat NK-1 receptor transfected on CHO cells using [125I]-Tyr] SP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed