Compile Data Set for Download or QSAR
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Found 3 Enz. Inhib. hit(s) with Target = 'Substance-P receptor' and Ligand = 'BDBM50049313'
TargetSubstance-P receptor(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50049313(2-Dimethylamino-N-{3-(1H-indol-3-yl)-2-[2-(4-pheny...)
Affinity DataIC50:  1.54nMAssay Description:Inhibitory activity against Tachykinin receptor 1 in human IM-9 cells using [125I]-labeled Boltan-Hunter substance P as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Mus musculus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50049313(2-Dimethylamino-N-{3-(1H-indol-3-yl)-2-[2-(4-pheny...)
Affinity DataIC50:  200nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1 in mouse brain using [125I]-labeled Boltan-Hunter substance P as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50049313(2-Dimethylamino-N-{3-(1H-indol-3-yl)-2-[2-(4-pheny...)
Affinity DataIC50:  480nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1 in rat brain using [125I]-labeled Boltan-Hunter substance P as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed