Compile Data Set for Download or QSAR
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Found 3 Enz. Inhib. hit(s) with Target = 'Substance-P receptor' and Ligand = 'BDBM50049338'
TargetSubstance-P receptor(GUINEA PIG)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50049338(CHEMBL353093 | N-[1-{[Acetyl-(2-methoxy-benzyl)-am...)
Affinity DataIC50:  0.880nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1 in guinea pig brain using [125I]-labeled Boltan-Hunter substance P as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50049338(CHEMBL353093 | N-[1-{[Acetyl-(2-methoxy-benzyl)-am...)
Affinity DataIC50:  0.880nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1 in guinea pig brain using [125I]-labeled Boltan-Hunter substance P as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50049338(CHEMBL353093 | N-[1-{[Acetyl-(2-methoxy-benzyl)-am...)
Affinity DataIC50:  16nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1 in rat brain using [125I]-labeled Boltan-Hunter substance P as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed