Compile Data Set for Download or QSAR
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Found 1 Enz. Inhib. hit(s) with Target = 'Substance-P receptor' and Ligand = 'BDBM50049348'
TargetSubstance-P receptor(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50049348(CHEMBL166240 | N-{1-(1H-Indol-3-ylmethyl)-2-[metha...)
Affinity DataIC50:  4nMAssay Description:Inhibitory activity against Tachykinin receptor 1 in human IM-9 cells using [125I]-labeled Boltan-Hunter substance P as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed