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Found 1 Enz. Inhib. hit(s) with Target = 'Substance-P receptor' and Ligand = 'BDBM50066219'
TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50066219((S)-1-(2-Fluoro-benzylthiocarbamoyl)-pyrrolidine-2...)
Affinity DataKi:  1.27E+3nMAssay Description:In vitro binding affinity towards Tachykinin receptor 1 to displace [3H][Sar9Met(O2)11]-SP (1 nM) binding to rabbit whole brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed