Compile Data Set for Download or QSAR
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Found 3 Enz. Inhib. hit(s) with Target = 'Substance-P receptor' and Ligand = 'BDBM50087852'
TargetSubstance-P receptor(Rattus norvegicus (rat))
Mississippi State University

Curated by ChEMBL
LigandPNGBDBM50087852(CHEMBL263185 | His-Asn-Pro-Ala-Ser-Phe-Ile-Gly-Leu...)
Affinity DataIC50:  32nMAssay Description:Displacement of [125I]Lys3-substance P from rat NK1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Marshall University School Of Medicine And Huntington Va Medical Center

Curated by ChEMBL
LigandPNGBDBM50087852(CHEMBL263185 | His-Asn-Pro-Ala-Ser-Phe-Ile-Gly-Leu...)
Affinity DataEC50:  13.5nMAssay Description:Agonist activity at bfSPR to produce increase in intracellular [Ca2+]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Marshall University School Of Medicine And Huntington Va Medical Center

Curated by ChEMBL
LigandPNGBDBM50087852(CHEMBL263185 | His-Asn-Pro-Ala-Ser-Phe-Ile-Gly-Leu...)
Affinity DataEC50:  14nMAssay Description:SP-induced [Ca2+] mobilization in CHO cells expressing human Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed