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Found 5 Enz. Inhib. hit(s) with Target = 'Substance-P receptor' and Ligand = 'BDBM50284050'
TargetSubstance-P receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50284050((S)-2-(2-Methoxy-phenyl)-1-((R)-1-oxo-4,4-diphenyl...)
Affinity DataIC50:  10nMAssay Description:Compound was evaluated for its affinity to rat Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50284050((S)-2-(2-Methoxy-phenyl)-1-((R)-1-oxo-4,4-diphenyl...)
Affinity DataIC50:  22.9nMAssay Description:Binding affinity was measured against the Tachykinin receptor 1 in human IM-9 cells using [3H]SP as ligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50284050((S)-2-(2-Methoxy-phenyl)-1-((R)-1-oxo-4,4-diphenyl...)
Affinity DataIC50:  49nMAssay Description:Compound was evaluated for its affinity, measured in [3H]-SP binding assay on human IM9 lymphoblast cultured cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50284050((S)-2-(2-Methoxy-phenyl)-1-((R)-1-oxo-4,4-diphenyl...)
Affinity DataIC50:  70nMAssay Description:Compound was evaluated for its affinity to guinea pig Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50284050((S)-2-(2-Methoxy-phenyl)-1-((R)-1-oxo-4,4-diphenyl...)
Affinity DataIC50:  70nMAssay Description:Compound was evaluated for its affinity to guinea pig Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails Article