Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Substance-P receptor' and Ligand = 'BDBM50327377'
TargetSubstance-P receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50327377((1S,2R,5aR,7S,8aS,8bS)-7-(benzylamino)-2-((R)-1-(3...)
Affinity DataIC50:  0.140nMAssay Description:Displacement of [125I]substance P from human NK1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50327377((1S,2R,5aR,7S,8aS,8bS)-7-(benzylamino)-2-((R)-1-(3...)
Affinity DataIC50:  2.30nMAssay Description:Displacement of [125I]substance P from human NK1 receptor expressed in CHO cells in presence of 50% human serumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed