Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) with Target = 'Substance-P receptor' and Ligand = 'BDBM50346326'
TargetSubstance-P receptor(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50346326((S)-2-acetyl-N-(3,5-bis(trifluoromethyl)benzyl)-N-...)
Affinity DataKd:  31.6nMAssay Description:Antagonist activity at human NK1 receptor expressed in CHO-K1 cells assessed as inhibition of substance P-induced calcium-dependent aequorine lumines...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2011
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50346326((S)-2-acetyl-N-(3,5-bis(trifluoromethyl)benzyl)-N-...)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]SP from human recombinant NK1 receptor expressed in CHO cells after 20 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2011
Entry Details Article
PubMed