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Found 3 Enz. Inhib. hit(s) with Target = 'Sucrase-isomaltase, intestinal' and Ligand = 'BDBM50024129'
TargetSucrase-isomaltase, intestinal(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50024129(5-Amino-1-hydroxymethyl-cyclohexane-1,2,3,4-tetrao...)
Affinity DataIC50:  49nMAssay Description:Alpha-D-glucosidase inhibitory activity and enzyme inhibition in vitro against porcine sucraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50024129(5-Amino-1-hydroxymethyl-cyclohexane-1,2,3,4-tetrao...)
Affinity DataIC50:  690nMAssay Description:Inhibition of rat intestinal brush border membrane sucraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50024129(5-Amino-1-hydroxymethyl-cyclohexane-1,2,3,4-tetrao...)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of rat intestinal brush border membrane isomaltaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed