Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with Target = 'TGF-beta receptor type-1' and Ligand = 'BDBM50015678'
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Ewha University—Industry Collaboration Foundation

US Patent
LigandPNGBDBM50015678(CHEMBL3260590 | USRE47141, Example 37)
Affinity DataIC50:  11.9nMAssay Description:ALK5 protein was expressed in Sf9 insect cells as human recombinant GST-fusion protein using the baculovirus expression system. Expressed protein was...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Ewha University—Industry Collaboration Foundation

US Patent
LigandPNGBDBM50015678(CHEMBL3260590 | USRE47141, Example 37)
Affinity DataIC50:  12nMAssay Description:Inhibition of human recombinant ALK5 expressed in insect Sf9 cells using casein as substrate by radioisotopic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Ewha University—Industry Collaboration Foundation

US Patent
LigandPNGBDBM50015678(CHEMBL3260590 | USRE47141, Example 37)
Affinity DataIC50:  1.46E+3nMAssay Description:Inhibition of human recombinant p38alpha expressed in Escherichia coli using ATF2 as substrate by radioisotopic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed