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Compile Data Set for Download or QSAR
maximum 50k data
Found
3
Enz. Inhib. hit(s) with Target = 'TGF-beta receptor type-2' and Ligand = 'BDBM283066'
Target
TGF-beta receptor type-2
(Homo sapiens (Human))
Rigel Pharmaceuticals
US Patent
Ligand
BDBM283066
(6-(1-(1-cyanocyclopropyl)-4-(4-fluorophenyl)-1H- i...)
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Affinity Data
IC50: 1.75E+3nM
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
UniProtKB/TrEMBL
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
TGF-beta receptor type-2
(Homo sapiens (Human))
Rigel Pharmaceuticals
US Patent
Ligand
BDBM283066
(6-(1-(1-cyanocyclopropyl)-4-(4-fluorophenyl)-1H- i...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 1.75E+3nM
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
UniProtKB/TrEMBL
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
TGF-beta receptor type-2
(Homo sapiens (Human))
Rigel Pharmaceuticals
US Patent
Ligand
BDBM283066
(6-(1-(1-cyanocyclopropyl)-4-(4-fluorophenyl)-1H- i...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 1.75E+3nM
Assay Description:
Assays for the compounds reported below were conducted in 1536-well plates and 2 mL reactions are prepared from addition of HIS-TGF-βR1 T204D or...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
UniProtKB/TrEMBL
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI