Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = 'Transient receptor potential cation channel subfamily V member 1' and Ligand = 'BDBM50155165'
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Purdue Pharma

Curated by ChEMBL
LigandPNGBDBM50155165(4-Pyridazin-3-yl-piperazine-1-carboxylic acid (4-i...)
Affinity DataIC50:  5.75E+3nMAssay Description:Inhibition of human vanilloid receptor 1 in HEK293 cells in capsaicin-induced FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Purdue Pharma

Curated by ChEMBL
LigandPNGBDBM50155165(4-Pyridazin-3-yl-piperazine-1-carboxylic acid (4-i...)
Affinity DataIC50:  1.33E+4nMpH: 5.5Assay Description:Inhibition of human vanilloid receptor 1 in HEK293 cells in pH 5.5-induced FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed