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Found 2 Enz. Inhib. hit(s) with Target = 'Transient receptor potential cation channel subfamily V member 1' and Ligand = 'BDBM50330643'
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50330643(CHEMBL1275621 | N-(4-tert-Butyl-benzyl)-2-(3-bromo...)
Affinity DataKi:  91nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50330643(CHEMBL1275621 | N-(4-tert-Butyl-benzyl)-2-(3-bromo...)
Affinity DataKi:  168nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells assessed as inhibition of capsaicin-induced calcium uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed