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Found 8 Enz. Inhib. hit(s) with Target = 'Translocator protein' and Ligand = 'BDBM50054125'
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50054125((E)-2-(2-(4-chlorophenyl)-1,2-dihydro-1-oxo-3H-pyr...)
Affinity DataIC50:  0.700nMAssay Description:Displacement of [3H]-PK11195 from rat kidney peripheral benzodiazepine receptor (type 1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50054125((E)-2-(2-(4-chlorophenyl)-1,2-dihydro-1-oxo-3H-pyr...)
Affinity DataIC50:  0.900nMAssay Description:Displacement of [3H]PK115 from peripheral benzodiazepine receptor in Sprague-Dawley rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50054125((E)-2-(2-(4-chlorophenyl)-1,2-dihydro-1-oxo-3H-pyr...)
Affinity DataIC50:  1.70nMAssay Description:Displacement of [3H]-Ro-5-4864 from rat kidney peripheral benzodiazepine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50054125((E)-2-(2-(4-chlorophenyl)-1,2-dihydro-1-oxo-3H-pyr...)
Affinity DataIC50:  1.90nMAssay Description:Binding affinity against peripheral benzodiazepine receptor( PBR).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50054125((E)-2-(2-(4-chlorophenyl)-1,2-dihydro-1-oxo-3H-pyr...)
Affinity DataIC50:  2.30nMAssay Description:Displacement of [3H]-Ro-5-4864 from rat cerebral cortex peripheral benzodiazepine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50054125((E)-2-(2-(4-chlorophenyl)-1,2-dihydro-1-oxo-3H-pyr...)
Affinity DataIC50:  9.80nMAssay Description:Displacement of [3H]-PK11195 from rat cerebral cortex peripheral benzodiazepine receptor (type 1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50054125((E)-2-(2-(4-chlorophenyl)-1,2-dihydro-1-oxo-3H-pyr...)
Affinity DataIC50:  14nMAssay Description:Displacement of [3H]-PK11195 from rat kidney peripheral benzodiazepine receptor (type 2)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50054125((E)-2-(2-(4-chlorophenyl)-1,2-dihydro-1-oxo-3H-pyr...)
Affinity DataIC50:  320nMAssay Description:Displacement of [3H]-PK11195 from rat cerebral cortex peripheral benzodiazepine receptor (type 2)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed