Compile Data Set for Download or QSAR
maximum 50k data
Found 8 Enz. Inhib. hit(s) with Target = 'Translocator protein' and Ligand = 'BDBM50054128'
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50054128(2-[2-(4-Chloro-phenyl)-1-oxo-1,2-dihydro-pyrrolo[3...)
Affinity DataIC50:  2.70nMAssay Description:Displacement of [3H]-PK11195 from rat kidney peripheral benzodiazepine receptor (type 1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50054128(2-[2-(4-Chloro-phenyl)-1-oxo-1,2-dihydro-pyrrolo[3...)
Affinity DataIC50:  4.90nMAssay Description:Displacement of [3H]-PK11195 from rat cerebral cortex peripheral benzodiazepine receptor (type 1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50054128(2-[2-(4-Chloro-phenyl)-1-oxo-1,2-dihydro-pyrrolo[3...)
Affinity DataIC50:  40nMAssay Description:Binding affinity against peripheral benzodiazepine receptor( PBR).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50054128(2-[2-(4-Chloro-phenyl)-1-oxo-1,2-dihydro-pyrrolo[3...)
Affinity DataIC50:  40nMAssay Description:Binding affinity against peripheral benzodiazepine receptor( PBR).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50054128(2-[2-(4-Chloro-phenyl)-1-oxo-1,2-dihydro-pyrrolo[3...)
Affinity DataIC50:  40nMAssay Description:Inhibition of rat liver Dihydrofolate reductase.More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50054128(2-[2-(4-Chloro-phenyl)-1-oxo-1,2-dihydro-pyrrolo[3...)
Affinity DataIC50:  120nMAssay Description:Displacement of [3H]-Ro-5-4864 from rat cerebral cortex peripheral benzodiazepine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50054128(2-[2-(4-Chloro-phenyl)-1-oxo-1,2-dihydro-pyrrolo[3...)
Affinity DataIC50:  160nMAssay Description:Displacement of [3H]-PK11195 from rat kidney peripheral benzodiazepine receptor (type 2)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50054128(2-[2-(4-Chloro-phenyl)-1-oxo-1,2-dihydro-pyrrolo[3...)
Affinity DataIC50:  210nMAssay Description:Displacement of [3H]-PK11195 from rat cerebral cortex peripheral benzodiazepine receptor (type 2)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed