Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with Target = 'Translocator protein' and Ligand = 'BDBM50509028'
TargetTranslocator protein(Homo sapiens (Human))
Macquarie University

Curated by ChEMBL
LigandPNGBDBM50509028(CHEMBL4161842)
Affinity DataKi:  70nMAssay Description:Displacement of [3H]PK11195 from wild-type human TSPO expressed in HEK293 cell membranes after 90 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Macquarie University

Curated by ChEMBL
LigandPNGBDBM50509028(CHEMBL4161842)
Affinity DataKi:  92nMAssay Description:Displacement of [3H]-PK11195 from wild type TSPO (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 90 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Macquarie University

Curated by ChEMBL
LigandPNGBDBM50509028(CHEMBL4161842)
Affinity DataKi:  319nMAssay Description:Displacement of [3H]PK11195 from human TSPO A147T mutant expressed in HEK293 cell membranes after 90 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Macquarie University

Curated by ChEMBL
LigandPNGBDBM50509028(CHEMBL4161842)
Affinity DataKi:  460nMAssay Description:Displacement of [3H]-PK11195 from TSPO A147T mutant (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 9...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed