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Found 3 Enz. Inhib. hit(s) with Target = 'Transporter' and Ligand = 'BDBM50019742'
TargetTransporter(Rattus norvegicus)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50019742(9-(3-((3S,5R)-3,5-dimethylpiperazin-1-yl)propyl)-9...)
Affinity DataKi:  2.16E+3nMAssay Description:Binding affinity at norepinephrine transporter using [3H]nisoxetine as radioligand from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50019742(9-(3-((3S,5R)-3,5-dimethylpiperazin-1-yl)propyl)-9...)
Affinity DataKi:  2.16E+3nMAssay Description:Displacement of [3H]nisoxetine from rat brain norepinephrine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50019742(9-(3-((3S,5R)-3,5-dimethylpiperazin-1-yl)propyl)-9...)
Affinity DataKi:  2.16E+3nMAssay Description:The compound was tested for binding affinity nisoxatine ligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed