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Found 5 Enz. Inhib. hit(s) with Target = 'Transporter' and Ligand = 'BDBM50127383'
TargetTransporter(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50127383(3-(4-Chloro-phenyl)-8-methyl-2-(3-phenyl-isoxazol-...)
Affinity DataKi:  220nMAssay Description:Binding affinity towards norepinephrine transporter was determined using [3H]nisoxetine radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50127383(3-(4-Chloro-phenyl)-8-methyl-2-(3-phenyl-isoxazol-...)
Affinity DataKi:  304nMAssay Description:Affinity for norepinephrine transporter determined by [3H]nisoxetine displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50127383(3-(4-Chloro-phenyl)-8-methyl-2-(3-phenyl-isoxazol-...)
Affinity DataIC50:  504nMAssay Description:Binding affinity towards Norepinephrine transporter was determined using NE[3H]Nisoxetine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50127383(3-(4-Chloro-phenyl)-8-methyl-2-(3-phenyl-isoxazol-...)
Affinity DataIC50:  504nMAssay Description:Inhibition of [3H]nisoxetine binding at norepinephrine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50127383(3-(4-Chloro-phenyl)-8-methyl-2-(3-phenyl-isoxazol-...)
Affinity DataIC50:  2.42E+3nMAssay Description:Inhibition of norepinephrine transporter (NET) determined using [3H]nisoxetine radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed