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Found 2 Enz. Inhib. hit(s) with Target = 'Tryptase beta-2' and Ligand = 'BDBM16310'
TargetTryptase beta-2(Homo sapiens (Human))
Arris

LigandPNGBDBM16310(2-(isoquinolin-3-yl)-1H-1,3-benzodiazole-6-carboxi...)
Affinity DataKi:  2.34E+4nMAssay Description:Enzymes were incubated with inhibitors at eight inhibitor concentrations bracketing the Ki, prepared by serial dilution along with control lacking th...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2(Homo sapiens (Human))
Arris

LigandPNGBDBM16310(2-(isoquinolin-3-yl)-1H-1,3-benzodiazole-6-carboxi...)
Affinity DataKi:  6.33E+4nM ΔG°:  -23.7kJ/molepH: 8.2 T: 2°CAssay Description:Enzymes were incubated with inhibitors at eight inhibitor concentrations bracketing the Ki, prepared by serial dilution along with control lacking th...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed