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Found 3 Enz. Inhib. hit(s) with Target = 'Tubulin alpha-1A chain' and Ligand = 'BDBM50106309'
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50106309(2-(2'-fluorophenyl)-6-pyrolinyl-4-(1H)-quinolone |...)
Affinity DataIC50:  457nMAssay Description:Inhibition of tubulin polymerization interacting at the colchicine binding site.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50106309(2-(2'-fluorophenyl)-6-pyrolinyl-4-(1H)-quinolone |...)
Affinity DataIC50:  7.60E+4nMAssay Description:Inhibition of colchicine binding(ICB). Tubulin concentration was 1 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50106309(2-(2'-fluorophenyl)-6-pyrolinyl-4-(1H)-quinolone |...)
Affinity DataIC50:  9.30E+4nMAssay Description:Inhibition of colchicine binding(ICB). [3H]-colchicine concentration was 5 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed