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Found 3 Enz. Inhib. hit(s) with Target = 'Tyrosine-protein kinase ABL1' and Ligand = 'BDBM50221548'
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Targegen

Curated by ChEMBL
LigandPNGBDBM50221548(4-(7-(1H-indol-4-yl)-5-methylbenzo[e][1,2,4]triazi...)
Affinity DataKi:  24nMAssay Description:Inhibition of AblMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Targegen

Curated by ChEMBL
LigandPNGBDBM50221548(4-(7-(1H-indol-4-yl)-5-methylbenzo[e][1,2,4]triazi...)
Affinity DataKi:  24nMAssay Description:Binding affinity to Abl (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Targegen

Curated by ChEMBL
LigandPNGBDBM50221548(4-(7-(1H-indol-4-yl)-5-methylbenzo[e][1,2,4]triazi...)
Affinity DataKi:  1.77E+3nMAssay Description:Binding affinity to Abl-T315I mutant (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed