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Found 2 Enz. Inhib. hit(s) with Target = 'Tyrosine-protein kinase ABL1 [1-999,Q252H]' and Ligand = 'BDBM68208'
TargetTyrosine-protein kinase ABL1 [1-999,Q252H](Homo sapiens (Human))
The Scripps Research Institute

LigandPNGBDBM68208(Type II inhibitor, 2)
Affinity DataIC50:  5nMpH: 7.5Assay Description:An in vitro kinase assay using dephophorylated conformationally inactive Abl kinase was obtained by treating pure recombinant Abl with Yersinia ester...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1 [1-999,Q252H](Homo sapiens (Human))
The Scripps Research Institute

LigandPNGBDBM68208(Type II inhibitor, 2)
Affinity DataIC50:  152nMpH: 7.5Assay Description:An in vitro kinase assay using phosphorylated recombinant human Abl kinase domains to phosphorylate a peptide substrate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed