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Found 3 Enz. Inhib. hit(s) with Target = 'Tyrosine-protein kinase BTK' and Ligand = 'BDBM50068543'
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM50068543(CHEMBL3402353)
Affinity DataIC50:  4.30nMAssay Description:Inhibition of biotinylated and unactivated BTK (unknown origin) using FITC-labeled Srctide peptide substrate and ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM50068543(CHEMBL3402353)
Affinity DataIC50:  189nMAssay Description:Inhibition of biotinylated and activated BTK (unknown origin) using FITC-labeled Srctide peptide substrate and ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM50068543(CHEMBL3402353)
Affinity DataKd:  5.5nMAssay Description:Binding affinity to biotinylated and unactivated BTK (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed